Gregory D. Vite : rechercher sur Z-Library

Vite, Gregory, Fraser-reid, Bert

Année:

2001

Langue:

english

Fichier:

PDF, 84 KB

english, 2001

Generation of Oxygen-Centered Radicals by Reaction of Nitrate Esters with Tri-n-Butyltin Hydride

Journal:

Synthetic Communications

Année:

1988

Langue:

english

Fichier:

PDF, 281 KB

english, 1988

Expedited mapping of the ligandable proteome using fully functionalized enantiomeric probe pairs

Wang, Yujia, Dix, Melissa M., Bianco, Giulia, Remsberg, Jarrett R., Lee, Hsin-Yu, Kalocsay, Marian, Gygi, Steven P., Forli, Stefano, Vite, Gregory, Lawrence, R. Michael, Parker, Christopher G., Cravat

Journal:

Nature Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.98 MB

english, 2019

Chemical Modification of Linkers Provide Stable Linker-payloads for the Generation of Antibody-drug Conjugates

Poudel, Yam B., Chowdari, Naidu S., Cheng, Heng, Iwuagwu, Christiana I., King, H. Dalton, Kotapati, Srikanth, Passmore, David, Rampulla, Richard, Mathur, Arvind, Vite, Gregory, Gangwar, Sanjeev

Journal:

ACS Medicinal Chemistry Letters

Année:

2020

Fichier:

PDF, 240 KB

2020

ChemInform Abstract: A Facile Method for the Transformation of N-(tert-Butoxycarbonyl) α-Amino Acids to N-Unprotected α-Amino Methyl Esters.

Bang-Chi Chen, Amanda P. Skoumbourdies, Peng Guo, Mark S. Bednarz, Octavian R. Kocy, Joseph E. Sundeen, Gregory D. Vite

Journal:

Année:

2000

Fichier:

PDF, 34 KB

2000

ChemInform Abstract: Synthesis, Structure Proof, and Biological Activity of Epothilone Cyclopropanes.

James Johnson, Soong-Hoon Kim, Marc Bifano, John DiMarco, Craig Fairchild, Jack Gougoutas, Francis Lee, Byron Long, John Tokarski, Gregory Vite

Journal:

Alicia Regueiro-Ren, Robert M. Borzilleri, Xiaoping Zheng, Soong-Hoon Kim, James A. Johnson, Craig R. Fairchild, Francis Y. F. Lee, Byron H. Long, Gregory D. Vite

Année:

2000

Fichier:

PDF, 31 KB

2000

ChemInform Abstract: Synthesis and Biological Activity of Novel Epothilone Aziridines.

Journal:

Année:

2001

Fichier:

PDF, 40 KB

2001

New dual inhibitors of EGFR and HER2 protein tyrosine kinases

Brian E. Fink, Gregory D. Vite, Harold Mastalerz, John F. Kadow, Soong-Hoon Kim, Kenneth J. Leavitt, Karen Du, Donald Crews, Toomas Mitt, Tai W. Wong, John T. Hunt, Dolatrai M. Vyas, John S. Tokarski

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 176 KB

english, 2005

Novel C-5 aminomethyl pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases

Harold Mastalerz, Ming Chang, Ashvinikumar Gavai, Walter Johnson, David Langley, Francis Y. Lee, Punit Marathe, Arvind Mathur, Simone Oppenheimer, James Tarrant, John S. Tokarski, Gregory D. Vite, Dol

Journal:

Année:

2007

Langue:

english

Fichier:

PDF, 293 KB

english, 2007

Identification of 2-amino-5-(thioaryl)thiazoles as inhibitors of nerve growth factor receptor TrkA

Soong-Hoon Kim, John S. Tokarski, Kenneth J. Leavitt, Brian E. Fink, Mark E. Salvati, Robert Moquin, Mary T. Obermeier, George L. Trainor, Gregory G. Vite, Linda K. Stadnick, Jonathan S. Lippy, Dan Yo

Journal:

Année:

2008

Langue:

english

Fichier:

PDF, 289 KB

english, 2008

Identification and optimization of a novel series of [2.2.1]-oxabicyclo imide-based androgen receptor antagonists

Mark E. Salvati, Aaron Balog, Weifang Shan, Richard Rampulla, Soren Giese, Tom Mitt, Joseph A. Furch, Gregory D. Vite, Ricardo M. Attar, Maria Jure-Kunkel, Jieping Geng, Cheryl A. Rizzo, Marco M. Gott

Journal:

Année:

2008

Langue:

english

Fichier:

PDF, 580 KB

english, 2008

Regioselective synthesis of folate receptor-targeted agents derived from epothilone analogs and folic acid

Iontcho R. Vlahov, Gregory D. Vite, Paul J. Kleindl, Yu Wang, Hari Krishna R. Santhapuram, Fei You, Stephen J. Howard, Soong-Hoon Kim, Francis F.Y. Lee, Christopher P. Leamon

Journal:

Année:

2010

Langue:

english

Fichier:

PDF, 467 KB

english, 2010

Novel pyrrolo[2,1-f][1,2,4]triazin-4-amines: Dual inhibitors of EGFR and HER2 protein tyrosine kinases

Brian E. Fink, Derek Norris, Harold Mastalerz, Ping Chen, Bindu Goyal, Yufen Zhao, Soong-Hoon Kim, Gregory D. Vite, Francis Y. Lee, Hongjian Zhang, Simone Oppenheimer, John S. Tokarski, Tai W. Wong, A

Journal:

Bert Fraser-Reid, Gregory D. Vite, Bik-Wah Anissa Yeung, Ray Tsang

Année:

2011

Langue:

english

Fichier:

PDF, 537 KB

english, 2011

On the question of reversibility in the intramolecular addition of radicals to aldehydes to form cycloalkanols

Journal:

Tetrahedron Letters

Année:

1988

Langue:

english

Fichier:

PDF, 205 KB

english, 1988

Optically active fluorinated cyclobutane nucleoside analogs with potent anti-herpes activity

Saleem Ahmad, Gregory S. Bisacchi, A.Kirk Field, Glenn A. Jacobs, A.Vickie Tuomari, Bridget McGeever-Rubin, Gregory D. Vite, Robert Zahler

Journal:

Cancer Chemotherapy and Pharmacology

Année:

1993

Langue:

english

Fichier:

PDF, 301 KB

english, 1993

Identification of novel functional inhibitors of 17β-hydroxysteroid dehydrogenase type III (17β-HSD3)

Thomas E. Spires, Brian E. Fink, Ellen K. Kick, Dan You, Cheryl A. Rizzo, Ivone Takenaka, R. Michael Lawrence, Zheming Ruan, Mark E. Salvati, Gregory D. Vite, Roberto Weinmann, Ricardo M. Attar, Marco

Journal:

The Prostate

Année:

2005

Langue:

english

Fichier:

PDF, 332 KB

english, 2005

Preclinical efficacy spectrum and pharmacokinetics of ixabepilone

Francis Y. F. Lee, Richard Smykla, Kathy Johnston, Krista Menard, Kelly McGlinchey, Russell W. Peterson, Amy Wiebesiek, Gregory Vite, Craig R. Fairchild, Robert Kramer

Journal:

Année:

2009

Langue:

english

Fichier:

PDF, 459 KB

english, 2009

Preclinical discovery of ixabepilone, a highly active antineoplastic agent

Francis Y. F. Lee, Robert Borzilleri, Craig R. Fairchild, Amrita Kamath, Richard Smykla, Robert Kramer, Gregory Vite

Journal:

Cancer Chemotherapy and Pharmacology

Année:

2008

Langue:

english

Fichier:

PDF, 451 KB

english, 2008

ChemInform Abstract: AlMe3-Promoted Formation of Amides from Acids and Amines.

Jianqing Li, Krishnananthan Subramaniam, Daniel Smith, Jennifer X. Qiao, Jie Jack Li, Jingfang Qian-Cutrone, John F. Kadow, Gregory D. Vite, Bang-Chi Chen

Journal:

Année:

2012

Fichier:

PDF, 41 KB

2012

A novel implanted device to wirelessly record and analyze continuous intracranial canine EEG

Kathryn A. Davis, Beverly K. Sturges, Charles H. Vite, Vanessa Ruedebusch, Gregory Worrell, Andrew B. Gardner, Kent Leyde, W. Douglas Sheffield, Brian Litt

Journal:

Epilepsy Research

Année:

2011

Langue:

english

Fichier:

PDF, 443 KB

english, 2011

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Discodermolide and Taxol: A Synergistic Drug Combination in Human Carcinoma Cell Lines

Année:

2001

Langue:

english

Fichier:

PDF, 1.26 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Some Recent Developments in the Synthesis and Structure-Activity Relationship of Novel Taxanes

Année:

2001

Langue:

english

Fichier:

PDF, 1.36 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Highly Efficient Semisynthesis of Biologically Active Epothilone Derivatives

Année:

2001

Langue:

english

Fichier:

PDF, 1.17 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || New Generation Taxoids and Hybrids of Microtuble-Stabilizing Anticancer Agents

Année:

2001

Langue:

english

Fichier:

PDF, 2.14 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Evolutionary Biosynthesis of Anticancer Drugs

Année:

2001

Langue:

english

Fichier:

PDF, 2.19 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Synthetic and Semisynthetic Analogs of Epothilones: Chemistry and Biological Activity

Année:

2001

Langue:

english

Fichier:

PDF, 1.41 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Farnesyltransferase Inhibitors as Potential Anticancer Agents

Année:

2001

Langue:

english

Fichier:

PDF, 811 KB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Synthesis and Biological Activity of Epothilones

Année:

2001

Langue:

english

Fichier:

PDF, 1.08 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Synthesis and Structure-Activity Relationship Studies of Cryptophycins: A Novel Class of Potent Antimitotic Antitumor Depsipeptides

Année:

2001

Langue:

english

Fichier:

PDF, 1.62 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Drugs to Enhance the Therapeutic Potency of Anticancer Antibodies: Antibody—Drug Conjugates as Tumor-Activated Prodrugs

Année:

2001

Langue:

english

Fichier:

PDF, 1.63 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Prospects for Antiangiogenic Therapies Based upon VEGF Inhibition

Année:

2001

Langue:

english

Fichier:

PDF, 1.77 MB

english, 2001

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Carbohydrate-Based Tumor Antigens as Antitumor Vaccine Agents

Année:

2001

Langue:

english

Fichier:

PDF, 1.43 MB

english, 2001

Synthesis, Structure Proof, and Biological Activity of Epothilone Cyclopropanes

Johnson, James, Kim, Soong-Hoon, Bifano, Marc, DiMarco, John, Fairchild, Craig, Gougoutas, Jack, Lee, Francis, Long, Byron, Tokarski, John, Vite, Gregory

Journal:

Alonso, Ricardo A., Burgey, Christopher S., Rao, B. Venkateswara, Vite, Gregory D., Vollerthun, Roland, Zottola, Mark A., Fraser-Reid, Bert

Année:

2000

Langue:

english

Fichier:

PDF, 155 KB

english, 2000

Carbohydrates to carbocycles: synthesis of the densely functionalized carbocyclic core of tetrodotoxin by radical cyclization of an anhydro sugar precursor

Journal:

Journal of the American Chemical Society

Année:

1993

Langue:

english

Fichier:

PDF, 963 KB

english, 1993

A practical, efficient large-scale synthesis of 1,6-anhydrohexopyranoses

Zottola, Mark A., Alonso, Ricardo, Vite, Gregory D., Fraser-Reid, Bert

Journal:

Année:

1989

Langue:

english

Fichier:

PDF, 465 KB

english, 1989

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Cancer Drug Discovery and Development: New Paradigms for a New Millennium

Regueiro-Ren, Alicia, Leavitt, Kenneth, Kim, Soong-Hoon, Höfle, Gerhard, Kiffe, Michael, Gougoutas, Jack Z., DiMarco, John D., Lee, Francis Y. F., Fairchild, Craig R., Long, Byron H., Vite, Gregory D.

Année:

2001

Langue:

english

Fichier:

PDF, 1.56 MB

english, 2001

SAR and pH Stability of Cyano-Substituted Epothilones

Journal:

Journal of Medicinal Chemistry

Année:

2002

Langue:

english

Fichier:

PDF, 197 KB

english, 2002

Discovery of the Pyrrolo[2,1- f ][1,2,4]triazine Nucleus as a New Kinase Inhibitor Template

Hunt, John T., Mitt, Toomas, Borzilleri, Robert, Gullo-Brown, Johnni, Fargnoli, Joseph, Fink, Brian, Han, Wen-Ching, Mortillo, Steven, Vite, Gregory, Wautlet, Barri, Wong, Tai, Yu, Chiang, Zheng, Xiao

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 62 KB

english, 2004

A Facile Method for the Transformation of N -( tert -Butoxycarbonyl) α-Amino Acids to N -Unprotected α-Amino Methyl Esters

Chen, Bang-Chi, Skoumbourdis, Amanda P., Guo, Peng, Bednarz, Mark S., Kocy, Octavian R., Sundeen, Joseph E., Vite, Gregory D.

Journal:

Perez, Heidi L., Cardarelli, Pina M., Deshpande, Shrikant, Gangwar, Sanjeev, Schroeder, Gretchen M., Vite, Gregory D., Borzilleri, Robert M.

Année:

1999

Langue:

english

Fichier:

PDF, 59 KB

english, 1999

Feasibility study of a caregiver seizure alert system in canine epilepsy

Coles, Lisa D., Patterson, Edward E., Sheffield, W. Douglas, Mavoori, Jaideep, Higgins, Jason, Michael, Bland, Leyde, Kent, Cloyd, James C., Litt, Brian, Vite, Charles, Worrell, Gregory A.

Journal:

Epilepsy Research

Année:

2013

Langue:

english

Fichier:

PDF, 1.00 MB

english, 2013

Antibody–drug conjugates: current status and future directions

Journal:

Drug Discovery Today

Année:

2014

Langue:

english

Fichier:

PDF, 876 KB

english, 2014

Pyrrolotriazine-5-carboxylate ester inhibitors of EGFR and HER2 protein tyrosine kinases and a novel one-pot synthesis of C-4 subsitituted pyrrole-2,3-dicarboxylate diesters

Mastalerz, Harold, Gavai, Ashvinikumar V, Fink, Brian, Struzynski, Charles, Tarrant, James, Vite, Gregory D, Wong, Tai W, Zhang, Guifen, Vyas, Dolatrai M

Journal:

Canadian Journal of Chemistry

Année:

2006

Fichier:

PDF, 93 KB

2006

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Pyrrolo[2,3- d ]pyrimidine and Pyrazolo[3,4- d ]pyrimidine Derivatives as Selective Inhibitors of the EGF Receptor Tyrosine Kinase

Li, Jianqing, Subramaniam, Krishnananthan, Smith, Daniel, Qiao, Jennifer X., Li, Jie Jack, Qian-Cutrone, Jingfang, Kadow, John F., Vite, Gregory D., Chen, Bang-Chi

Année:

2001

Langue:

english

Fichier:

PDF, 1.29 MB

english, 2001

AlMe 3 -Promoted Formation of Amides from Acids and Amines

Journal:

Vite, Gregory D., Spencer, Thomas A.

Année:

2012

Langue:

english

Fichier:

PDF, 287 KB

english, 2012

Exploration of a novel cyclization reaction. Synthesis of (.+-.)-.beta.-eudesmol

Journal:

Vite, Gregory D., Alonso, Ricardo, Fraser-Reid, Bert

Année:

1988

Langue:

english

Fichier:

PDF, 867 KB

english, 1988

Intramolecular radical cyclizations of 2-deoxy-2-iodohexopyranoside derivatives: routes to densely functionalized carbocycles

Journal:

Journal of Medicinal Chemistry

Année:

1989

Langue:

english

Fichier:

PDF, 379 KB

english, 1989

Development of Highly Potent Inhibitors of Ras Farnesyltransferase Possessing Cellular and in Vivo Activity

Leftheris, Katerina, Kline, Toni, Vite, Gregory D., Cho, Young H., Bhide, Rajeev S., Patel, Dinesh V., Patel, Manorama M., Schmidt, Robert J., Weller, Harold N., Andahazy, Mary L., Carboni, Joan M., G

Journal:

Année:

1996

Langue:

english

Fichier:

PDF, 415 KB

english, 1996

Synthesis of (.+-.)-7-epivaleranone and (.+-.)-valeranone

Vite, Gregory D., Spencer, Thomas A.

Journal:

Yeung, Bik-Wah Anissa, Alonso, Ricardo, Vite, Gregory D., Fraser-reid, Bert

Année:

1988

Langue:

english

Fichier:

PDF, 906 KB

english, 1988

Carbohydrates to Carbocycles via Radical Aldehyde Cyclizations

Journal:

Journal of Carbohydrate Chemistry

Année:

1989

Langue:

english

Fichier:

PDF, 679 KB

english, 1989

[ACS Symposium Series] Anticancer Agents Volume 796 (Frontiers in Cancer Chemotherapy) || Inhibiting Fornesyl Protein Transferase with Sch-66336: Potentially a Selective, Noncytotoxic Therapy for Human Cancer